Solid pharmaceutical compositions comprising a SIP receptor agonist and a sugar alcohol
DC CAFC
First Claim
Patent Images
1. A solid pharmaceutical composition suitable for oral administration, comprising:
- (a) a S1P receptor agonist which is selected from 2-amino-2-[4-(3-benzyloxyphenoxy)-2-chlorophenyl]propyl-1,3-propane-diol or 2-amino-2-[4-(3-benzyloxyphenylthio)-2-chlorophenyl]propyl-1,3-propane-diol, 2-amino-2-[4-(3-benzyloxyphenylthio)-2-chlorophenyl]-2-ethyl-1,3-propane-diol, and its phosphates or a pharmaceutically acceptable salt thereof; and
(b) a sugar alcohol.
1 Assignment
Litigations
2 Petitions
Accused Products
Abstract
A solid pharmaceutical composition suitable for oral administration, comprising:
- (a) a S1P receptor agonist; and
- (b) a sugar alcohol.
12 Citations
32 Claims
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1. A solid pharmaceutical composition suitable for oral administration, comprising:
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(a) a S1P receptor agonist which is selected from 2-amino-2-[4-(3-benzyloxyphenoxy)-2-chlorophenyl]propyl-1,3-propane-diol or 2-amino-2-[4-(3-benzyloxyphenylthio)-2-chlorophenyl]propyl-1,3-propane-diol, 2-amino-2-[4-(3-benzyloxyphenylthio)-2-chlorophenyl]-2-ethyl-1,3-propane-diol, and its phosphates or a pharmaceutically acceptable salt thereof; and (b) a sugar alcohol. - View Dependent Claims (2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 32)
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- 19. A solid pharmaceutical composition suitable for oral administration, comprising mannitol and 2-amino-2-[2-(4-octylphenyl)ethyl]propane-1,3-diol or a pharmaceutically acceptable salt thereof.
Specification
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Litigation Data
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Current AssigneeMitsubishi Tanabe Pharma Corporation (Mitsubishi Chemical Group Corp.), Novartis Ag
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Original AssigneeMitsubishi Tanabe Pharma Corporation (Mitsubishi Chemical Group Corp.), Novartis Ag
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InventorsOomura, Tomoyuki, Pudipeddi, Madhusudhan, Ruegger, Colleen, Sasaki, Masaki, Tamura, Tokuhiro, Royce, Alan E
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Primary Examiner(s)PACKARD, BENJAMIN J
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Application NumberUS12/189,323Publication NumberTime in Patent Office1,576 DaysField of Search514/649US Class Current514/649CPC Class CodesA61K 2300/00 Mixtures or combinations of...A61K 31/135 having aromatic rings , e.g...A61K 31/137 Arylalkylamines, e.g. amphe...A61K 31/138 Aryloxyalkylamines, e.g. pr...A61K 31/145 having sulfur, e.g. thiuram...A61K 45/06 Mixtures of active ingredie...A61K 47/10 Alcohols; Phenols; Salts th...A61K 47/26 Carbohydrates, e.g. sugar a...A61K 9/0053 Mouth and digestive tract, ...A61K 9/2013 Organic compounds, e.g. pho...A61K 9/2018 Sugars, or sugar alcohols, ...A61K 9/2054 Cellulose; Cellulose deriva...A61K 9/4858 Organic compoundsA61K 9/4866 Organic macromolecular comp...A61P 25/00 Drugs for disorders of the ...A61P 25/28 for treating neurodegenerat...A61P 29/00 Non-central analgesic, anti...A61P 31/00 Antiinfectives, i.e. antibi...A61P 31/12 AntiviralsA61P 37/00 Drugs for immunological or ...View All
